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Member
- Apr 8, 2020
- 62
While looking for sources I discovered a russian drug "Tiapride" (Tiapridal) which is avaliable at an online shop.
It was never mentioned here but it looked promising as an anti emetic
It also blocks D3 recepters and acts as sedative. Could we be killing two birds with one stone here and be using this as an anticonvulsant as well aas an antiemetic? It was never mentioned anywhere and its getting hard to find other antiemetics so i thought i would share it. Perhaps someone has had experience with this drug?
It was never mentioned here but it looked promising as an anti emetic
Tiapride is a drug that selectively blocks D2 and D3 dopamine receptors in the brain. It is used to treat a variety of neurological and psychiatric disorders including dyskinesia, alcohol withdrawal syndrome, negative symptoms of psychosis, and agitation and aggression in the elderly.[1] A derivative of benzamide, tiapride is chemically and functionally similar to other benzamide antipsychotics such as sulpiride and amisulpride known for their dopamine antagonist effects.
TIAPRIDE (Tiapridal) is a neuroleptic that has hypnotic, sedative, analgesic effects. It provides sedative, antiemetic and hypothermic action by blocking adrenergic, dopamine and dopamine D 2-receptors in the brain. Tiapride is used to treat psychomotor agitation and aggressive states, especially in chronic alcoholism, dyskinesia, alcohol withdrawal syndrome. Due to antagonistic effect on striatal dopamine receptors it is effective in treating motor deficits, such as tardive dyskinesia and chorea.
It also blocks D3 recepters and acts as sedative. Could we be killing two birds with one stone here and be using this as an anticonvulsant as well aas an antiemetic? It was never mentioned anywhere and its getting hard to find other antiemetics so i thought i would share it. Perhaps someone has had experience with this drug?